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Oral Angiotensin-Converting Enzyme (ACE) Inhibitors and Angiotensin II Receptor Blockers for Hypertension

Medication

Selected Adverse Effects

ACE inhibitors*

BenazeprilBenazepril

Rash, cough, angioedema, hyperkalemia (particularly in patients with renal insufficiency or taking nonsteroidal anti-inflammatory drugs, potassium-sparing diuretics, or potassium supplements), dysgeusia, reversible acute kidney injury if stenosis affecting one or both kidneys threatens renal function, proteinuria (rare at recommended doses), neutropenia (rare), hypotension with initiation of treatment (particularly in patients with high plasma renin activity or with hypovolemia due to diuretics or other conditions)

CaptoprilCaptopril

EnalaprilEnalapril

FosinoprilFosinopril

LisinoprilLisinopril

PerindoprilPerindopril

QuinaprilQuinapril

RamiprilRamipril

TrandolaprilTrandolapril

Angiotensin II receptor blockers

AzilsartanAzilsartan

Dizziness, angioedema (very rare); theoretically, same adverse effects as ACE inhibitors on renal function (except proteinuria and neutropenia), serum potassium, and blood pressure

CandesartanCandesartan

Eprosartan

IrbesartanIrbesartan

LosartanLosartan

OlmesartanOlmesartan

TelmisartanTelmisartan

ValsartanValsartan

* All ACE inhibitors and angiotensin II receptor blockers are contraindicated in pregnancy (can cause injury or death to the developing fetus).