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Some Medications That Cause Immunosuppression

Class

Examples

Antiseizure medications

LamotrigineLamotrigine

PhenytoinPhenytoin

Valproate

Biologics and small molecules

Interleukin (IL)-1 inhibitors (eg, anakinra)Interleukin (IL)-1 inhibitors (eg, anakinra)

IL-6 inhibitors (eg, tocilizumab)IL-6 inhibitors (eg, tocilizumab)

IL-17 inhibitors (eg, brodalumab)IL-17 inhibitors (eg, brodalumab)

Tumor necrosis factor (TNF) inhibitors (eg, adalimumab, etanercept, infliximab)Tumor necrosis factor (TNF) inhibitors (eg, adalimumab, etanercept, infliximab)

T-cell activation inhibitors (eg, abatacept, basiliximab)T-cell activation inhibitors (eg, abatacept, basiliximab)

CD20 inhibitors (eg, rituximab, ofatumumab)CD20 inhibitors (eg, rituximab, ofatumumab)

CD3 inhibitors (eg, muromonab-CD3)

Complement inhibitors (eg, sutimlimab, pegcetacoplan, eculizumab, avacopan) Complement inhibitors (eg, sutimlimab, pegcetacoplan, eculizumab, avacopan)

Janus kinase (JAK) inhibitors (eg, ruxolitinib)Janus kinase (JAK) inhibitors (eg, ruxolitinib)

Other B cell–targeting medications (eg, blinatumomab, belimumab, axicabtagene ciloleucel [CART-T therapy])Other B cell–targeting medications (eg, blinatumomab, belimumab, axicabtagene ciloleucel [CART-T therapy])

Calcineurin inhibitors

CyclosporineCyclosporine

TacrolimusTacrolimus

VoclosporinVoclosporin

Corticosteroids

MethylprednisoloneMethylprednisolone

PrednisonePrednisone

Cytotoxic chemotherapy agents

Multiple (see Systemic Antineoplastic Therapy)

Immunosuppressive immunoglobulins

Antilymphocyte globulin

Antithymocyte globulinAntithymocyte globulin

Purine metabolism inhibitors

AzathioprineAzathioprine

MycophenolateMycophenolate

Rapamycins

EverolimusEverolimus

SirolimusSirolimus